Next Era PeptideNext Era Peptide

MOTS-C

Mitochondrial Open Reading Frame of the 12S rRNA-c

Molecular Details

SequenceMet-Arg-Trp-Gln-Glu-Met-Gly-Tyr-Ile-Phe-Tyr-Pro-Arg-Lys-Leu-Arg
Molecular FormulaC₁₀₁H₁₅₂N₂₈O₂₂S₂
Molecular Weight2,174.6 Da
CAS Number1627580-64-6

Overview

MOTS-c is a 16-amino acid mitochondrial-derived peptide (MDP) encoded by the mitochondrial MT-RNR1 gene rather than the nuclear genome. Discovered in 2015, it represents a unique class of bioactive compounds derived from organellar genomes. The peptide is activated by metabolic stress and physical exercise, with expression declining with age. MOTS-c signals through the folate-AICAR-AMPK pathway, and is the first mitochondrial-encoded peptide to advance into human clinical trials.

Published Research

Metabolic Homeostasis & Obesity

In vivo (mouse) · 2015

The seminal discovery study published in Cell Metabolism showed MOTS-c administration reduces obesity and insulin resistance in mouse models through AMPK-dependent pathways and enhanced glucose utilization in skeletal muscle.

Type 2 Diabetic Cardiac Function

In vivo (rat) · 2025

In diabetic rat models, daily MOTS-c administration for 3 weeks restored mitochondrial respiration, improved cardiac contractility, and upregulated antioxidant defense genes (catalase, SOD2).

Pancreatic Islet Senescence Prevention

In vivo (aging mice) · 2025

MOTS-c treatment reduced age-related pancreatic islet cell senescence, improved glucose tolerance, and delayed progression of diabetes in aging mice through mitochondrial function enhancement.

Anti-inflammatory & Analgesic Mechanism

In vivo (mouse) · 2020

MOTS-c administration produced antinociceptive and anti-inflammatory effects via AMPK pathway activation in formalin-induced pain models, linking mitochondrial peptide signaling to neuroinflammatory processes.

Storage & Handling

Store lyophilized powder at –20°C or –80°C. Contains methionine — vulnerable to oxidative degradation; nitrogen or argon purging recommended. Prepare solutions fresh and aliquot for immediate use. Avoid repeated freeze-thaw cycles.

For research purposes only. Not intended for human consumption. This profile summarizes published preclinical literature and does not constitute medical, clinical, or dosage guidance.